Synonyms
Taltirelin Acetate
Ceredist
TA 0910
Description
Taltirelin is a thyrotropin-releasing hormone receptor (TRH-R) superagonist with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Molecular Formula
C17H23N7O5
SMILES
CN1C(=O)CC(NC1=O)C(=O)NC(CC2=CN=CN2)C(=O)N3CCCC3C(=O)N
Density, g/cm3
1.447±0.06 (Predicted)